平安! 发表于 2011-11-9 19:57 / e' T* i. g3 n, F) q9 e
Pazopanib (100 mg/kg/day free base equivalent)
]' w. f6 X3 X2 \" d 这是个已经在美国上市的老药了,能下载到正式药物使用说明书英文版。
( d `/ X0 V! v2 L搜索了一下,原料一大堆。3 @7 \1 ^$ J9 p6 H/ j! Z
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对不起!100mg/kg是用于移植瘤的,我弄错了。1 |4 P* @' F% n
# g/ E" R7 \* j& ~, u0 P& P/ O以下是正版说明书的推荐用量。9 [2 ^0 ~+ h3 S% C4 g0 h
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--------------------- DOSAGE AND ADMINISTRATION ----------------$ f4 ^/ \6 s* I$ ~
* 800 mg orally once daily without food (at least 1 hour before or 2 hours after a meal). (2.1) + ?( V$ c! V6 t
* Baseline moderate hepatic impairment – 200 mg orally once daily. Not recommended in patients with severe hepatic impairment. (2.2) 8 V0 @5 E+ b* T' |1 e- N: _
---------------------DOSAGE FORMS AND STRENGTHS --------------; c! d* b, j0 u2 Z+ w5 R9 ]
200 mg tablets. (3)
2 N' e0 S1 `3 b$ K-------------------------------CONTRAINDICATIONS------------------------ |